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Projekt Druckansicht

Ortsspezifisches Crosslinking mit KLK-Proteasen aus Prostata

Fachliche Zuordnung Biologische und Biomimetische Chemie
Förderung Förderung von 2019 bis 2023
Projektkennung Deutsche Forschungsgemeinschaft (DFG) - Projektnummer 409661645
 
Erstellungsjahr 2024

Zusammenfassung der Projektergebnisse

This project focused on improving and designing new orthogonal components for protein translation with "clickable" noncanonical amino acids (ncAAs) to create molecular tools for bioconjugation. Human kallikrein-related peptidases (KLKs), involved in fertilization and prostate cancer, were selected as the model proteins. The goal was to apply Selective Pressure Incorporation (SPI) and Stop Codon Suppression (SCS) methods in KLK studies. While SPI is well-established, especially with "clickable" ncAAs, the orthogonal translation system achieved a breakthrough by efficiently incorporating more than 20 ncAAs into model proteins. These ncAAs, containing small bioorthogonal tags, are ideal for various click chemistry applications. Additionally, system efficiency was significantly improved by introducing solubility tags to enhance enzyme folding and utilizing translational components from psychrophilic (cold-adapted) organisms for enhanced performance ("cold" orthogonal translation).

Projektbezogene Publikationen (Auswahl)

 
 

Zusatzinformationen

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